Regular paperTargetability of novel immunoliposomes modified with amphipathic poly(ethylene glycol) s conjugated at their distal terminals to monoclonal antibodies
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Keywords
Liposome
Immunoliposome
Antibody
Poly(ethylene glycol)
Drug delivery system
Abbreviations
CH, cholesterol
DF, deferoxamine
DSPE, distearoyl phosphatidylethanolamine
DSPE-PEG, distearoyl-N-(monomethoxy poly(ethylene glycol) succinyl)phosphatidylethanolamine
DSPE-PEG-COOH, distearoyl-N-(3-carboxypropionoyl poly(ethylene glycol) succinyl)phosphatidylethanolamine
ePC, egg phosphatidylcholine
Mes, 2-(N-morpholino)ethanesulfonic acid hemisodium salt
NGPE, N-glutaryldistearoylphosphatidylethanolamine
PEG-OSu, monomethoxy poly(ethylene glycol) succinimidyl succinate
PEG-2)Su, poly(ethylene glycol) bis(succinimidyl succinate)
SUV, small unilamellar vesicle
34A, rat monoclonal IgG2a antibody
14, rat monoclonal IgG2a antibody, a subtype-matched nonspecific control antibody to 34A
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Copyright © 1995 Published by Elsevier B.V.